• 产品编号:Asc-576
    • 产品名称:Asenapine maleate
    • 产品规格:10mg/50mg
    • 价  格:611.00/2498.00
    • 供 应 商:Ascent
    • 库  存:
  • Product name

    Asenapine maleate

    Description

    Multiple receptor antagonist. Anti-psychotic agent.

    Alternative names

    • ASE

    Biological description

    Novel, multiple receptor antagonist. Displays activity at 5-HT, dopamine, adrenoceptors and histamine receptors. (pKi values are 8.60 (5-HT1A), 8.40 (5-HT1B), 10.15 (5-HT2A), 9.75 (5-HT2B), 10.46 (5-HT2C), 8.84 (5-HT5A), 9.60 (5-HT6), 9.94 (5-HT7), 8.85 (D1), 8.90 (D2L), 8.84 (D2S), 9.38 (D3), 8.95 (D4), 8.93 (a1A), 8.9 (a2A), 9.49 (a2B), 8.91 (a2C), 9.00 (H1) and 8.21(H2) receptors respectively). Increases dopamine, norepinephrine and acetylcholine efflux. Anti-psychotic in vivo.

    Purity

    > 99%

    General notes

    Providing storage is as stated on the product vial and the vial is kept tightly sealed, the product can be stored for up to 6 months.

    Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour.

    Properties

    Chemical name

    trans-5-Chloro-2-methyl-2,3,3a,12b-tetrahydro-1H-dibenzo[2,3:6,7]oxepino[4,5-c]pyrrole maleate

    Molecular Weight

    401.85

    Chemical structure

    Chemical Structure

    Molecular formula

    C17H16ClNO.C4H4O4

    CAS Number

    85650-56-2

    Solubility

    Soluble in DMSO to 100 mM and in ethanol to 100 mM

    Storage instructions

    Store at +4°C.

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